Summary of all-grade nonhematologic adverse events occurring in >10% of patients and all treatment-emergent hematologic adverse events
| Toxicity . | Grade 1/2, n (%) . | Grade 3, n (%) . | Grade 4, n (%) . | Total, n (%) . |
|---|---|---|---|---|
| Nonhematologic | ||||
| Fatigue | 10 (36) | 2 (7.1) | 0 | 12 (43) |
| Rash | 7 (25) | 1 (3.6) | 0 | 8 (29) |
| Transaminitis | 6 (21) | 2 (7.1) | 0 | 8 (29) |
| Fever | 4 (14) | 1 (3.6) | 0 | 5 (18) |
| Lipase elevation | 1 (3.6) | 2 (7.1) | 2 (7.1) | 5 (18) |
| Pneumonitis | 3 (11) | 1 (3.6) | 0 | 4 (14) |
| Abdominal pain | 3 (11) | 1 (3.6) | 0 | 4 (14) |
| Nausea | 3 (11) | 1 (3.6) | 0 | 4 (14) |
| Vomiting | 4 (14) | 0 | 0 | 4 (14) |
| Arthralgia | 2 (7.1) | 1 (3.6) | 0 | 3 (11) |
| Bilirubin increase | 0 | 3 (11) | 0 | 3 (11) |
| Confusion | 2 (7.1) | 1 (3.6) | 0 | 3 (11) |
| Diarrhea | 3 (11) | 0 | 0 | 3 (11) |
| Dry mouth | 3 (11) | 0 | 0 | 3 (11) |
| Headache | 3 (11) | 0 | 0 | 3 (11) |
| Hematologic | ||||
| Thrombocytopenia | 2 (7.1) | 0 | 4 (14) | 6 (21) |
| Neutropenia | 1 (3.6) | 1 (3.6) | 3 (11) | 5 (18) |
| Anemia | 1 (3.6) | 3 (11) | 0 | 4 (14) |
| Febrile neutropenia | 0 | 2 (7.1) | 1 (3.6) | 3 (11) |
| Toxicity . | Grade 1/2, n (%) . | Grade 3, n (%) . | Grade 4, n (%) . | Total, n (%) . |
|---|---|---|---|---|
| Nonhematologic | ||||
| Fatigue | 10 (36) | 2 (7.1) | 0 | 12 (43) |
| Rash | 7 (25) | 1 (3.6) | 0 | 8 (29) |
| Transaminitis | 6 (21) | 2 (7.1) | 0 | 8 (29) |
| Fever | 4 (14) | 1 (3.6) | 0 | 5 (18) |
| Lipase elevation | 1 (3.6) | 2 (7.1) | 2 (7.1) | 5 (18) |
| Pneumonitis | 3 (11) | 1 (3.6) | 0 | 4 (14) |
| Abdominal pain | 3 (11) | 1 (3.6) | 0 | 4 (14) |
| Nausea | 3 (11) | 1 (3.6) | 0 | 4 (14) |
| Vomiting | 4 (14) | 0 | 0 | 4 (14) |
| Arthralgia | 2 (7.1) | 1 (3.6) | 0 | 3 (11) |
| Bilirubin increase | 0 | 3 (11) | 0 | 3 (11) |
| Confusion | 2 (7.1) | 1 (3.6) | 0 | 3 (11) |
| Diarrhea | 3 (11) | 0 | 0 | 3 (11) |
| Dry mouth | 3 (11) | 0 | 0 | 3 (11) |
| Headache | 3 (11) | 0 | 0 | 3 (11) |
| Hematologic | ||||
| Thrombocytopenia | 2 (7.1) | 0 | 4 (14) | 6 (21) |
| Neutropenia | 1 (3.6) | 1 (3.6) | 3 (11) | 5 (18) |
| Anemia | 1 (3.6) | 3 (11) | 0 | 4 (14) |
| Febrile neutropenia | 0 | 2 (7.1) | 1 (3.6) | 3 (11) |