Table 1.

RXR-specific ligand LG100268 enhances CDDO-Me-induced apoptosis in HL-60 cells (24 hours)

LG100268CDDO-Me
00.1 μM
4.4 22.4 
10 nM 6.8 34.4  
100 nM 6.2 40.3 
1 μM 6.3 61.6 
LG100268CDDO-Me
00.1 μM
4.4 22.4 
10 nM 6.8 34.4  
100 nM 6.2 40.3 
1 μM 6.3 61.6 

Results are expressed as a percentage of sub-G1 cells (flow cytometry).

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