Treatment-emergent AEs occurring in at least 2 patients regardless of attribution
| . | n (%) . | ||||
|---|---|---|---|---|---|
| 100 mg (n = 6) . | 150 mg (n = 6) . | Total (N = 12) . | |||
| Grade 1/2 . | Grade 3 . | Grade 1/2 . | Grade 3 . | All grades . | |
| Diarrhea | 5 (83.3) | 1 (16.7) | 5 (83.3) | 11 (91.7) | |
| Fatigue | 4 (66.7) | 2 (33.3) | 3 (50.0) | 1 (16.7) | 10 (83.3) |
| Constipation | 6 (100) | 4 (66.7) | 10 (83.3) | ||
| Nausea | 5 (83.3) | 5 (83.3) | 10 (83.3) | ||
| Headache | 4 (66.7) | 1 (16.7) | 2 (33.3) | 7 (50) | |
| Abdominal pain | 4 (66.7) | 2 (33.3) | 6 (50) | ||
| Upper respiratory tract infection | 1 (16.7) | 4 (66.7) | 5 (41.7) | ||
| Dry skin | 2 (33.3) | 2 (33.3) | 4 (33.3) | ||
| Pain | 2 (33.3) | 1 (16.7) | 1 (16.7) | 4 (33.3) | |
| Pruritus | 2 (33.3) | 2 (33.3) | 4 (33.3) | ||
| Vomiting | 3 (50.0) | 1 (16.7) | 4 (33.3) | ||
| Arthralgia | 3 (50) | 3 (25) | |||
| Dizziness | 3 (50) | 3 (25) | |||
| Cough | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Decreased appetite | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Dyspepsia | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Flushing | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Oropharyngeal pain | 1 (16.7) | 2 (33.3) | 3 (25.0) | ||
| Dysgeusia | 1 (16.7) | 2 (33.3) | 3 (25.0) | ||
| Dyspepsia | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Epistaxis | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Weight gain | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Alopecia | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Anorexia | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Back pain | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Chest pain | 2 (33.3) | 2 (16.7) | |||
| Disorientation | 2 (33.3) | 2 (16.7) | |||
| Eye infection | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Flatulence | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| GERD | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Heartburn | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Rash | 2 (33.3) | 2 (16.7) | |||
| Sinusitis | 2 (16.7) | 2 (16.7) | |||
| . | n (%) . | ||||
|---|---|---|---|---|---|
| 100 mg (n = 6) . | 150 mg (n = 6) . | Total (N = 12) . | |||
| Grade 1/2 . | Grade 3 . | Grade 1/2 . | Grade 3 . | All grades . | |
| Diarrhea | 5 (83.3) | 1 (16.7) | 5 (83.3) | 11 (91.7) | |
| Fatigue | 4 (66.7) | 2 (33.3) | 3 (50.0) | 1 (16.7) | 10 (83.3) |
| Constipation | 6 (100) | 4 (66.7) | 10 (83.3) | ||
| Nausea | 5 (83.3) | 5 (83.3) | 10 (83.3) | ||
| Headache | 4 (66.7) | 1 (16.7) | 2 (33.3) | 7 (50) | |
| Abdominal pain | 4 (66.7) | 2 (33.3) | 6 (50) | ||
| Upper respiratory tract infection | 1 (16.7) | 4 (66.7) | 5 (41.7) | ||
| Dry skin | 2 (33.3) | 2 (33.3) | 4 (33.3) | ||
| Pain | 2 (33.3) | 1 (16.7) | 1 (16.7) | 4 (33.3) | |
| Pruritus | 2 (33.3) | 2 (33.3) | 4 (33.3) | ||
| Vomiting | 3 (50.0) | 1 (16.7) | 4 (33.3) | ||
| Arthralgia | 3 (50) | 3 (25) | |||
| Dizziness | 3 (50) | 3 (25) | |||
| Cough | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Decreased appetite | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Dyspepsia | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Flushing | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Oropharyngeal pain | 1 (16.7) | 2 (33.3) | 3 (25.0) | ||
| Dysgeusia | 1 (16.7) | 2 (33.3) | 3 (25.0) | ||
| Dyspepsia | 2 (33.3) | 1 (16.7) | 3 (25.0) | ||
| Epistaxis | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Weight gain | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Alopecia | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Anorexia | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Back pain | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Chest pain | 2 (33.3) | 2 (16.7) | |||
| Disorientation | 2 (33.3) | 2 (16.7) | |||
| Eye infection | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Flatulence | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| GERD | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Heartburn | 1 (16.7) | 1 (16.7) | 2 (16.7) | ||
| Rash | 2 (33.3) | 2 (16.7) | |||
| Sinusitis | 2 (16.7) | 2 (16.7) | |||
GERD, gastroesophageal reflux disease.