Table 1

Inhibitory concentrations of EXEL-0862 against several protein tyrosine kinases

KinaseIC50, nM
KIT 8.5 
KIT D816V 42 
PDGFRβ 1.1 
VEGFR2 2.0 
FGFR1 4.0 
FLT3 1.5 
InsulinR 1603 
KinaseIC50, nM
KIT 8.5 
KIT D816V 42 
PDGFRβ 1.1 
VEGFR2 2.0 
FGFR1 4.0 
FLT3 1.5 
InsulinR 1603 
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