Table 1. In vitro enzymatic IC 50 values... | American Society of Hematology

Table 1.

In vitro enzymatic IC₅₀ values of different PI3K inhibitors on class I PI3Ks

	In vitro IC₅₀, μM
Inhibitor	p110α	p110β	p110δ	p110γ
IC87114	> 100	1.82	0.07	1.24
LY294002	0.7	0.306	1.33	7.26
AS-604850	3.4	> 20	> 20	0.19

	In vitro IC₅₀, μM
Inhibitor	p110α	p110β	p110δ	p110γ
IC87114	> 100	1.82	0.07	1.24
LY294002	0.7	0.306	1.33	7.26
AS-604850	3.4	> 20	> 20	0.19