Urine excretion of dGuo and inosine after a single intravenous infusion of forodesine
. | . | . | Urine dGuo . | . | . | Urine inosine . | . | . | ||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Patient no. . | Dose, mg/m2 . | Dose, mg . | Amount excreted, mg . | Tmax, h . | Maximum rate, mg/h . | Amount excreted, mg . | Tmax, h . | Maximum rate, mg/h . | ||||
| 1 | 40 | 79.2 | 213.9 | 16 | 11.5 | 1151.5 | 16 | 59.8 | ||||
| 2 | 40 | 67.2 | 95.1 | 16 | 4.8 | 578.1 | 16 | 29.9 | ||||
| 3 | 40 | 64.4 | 172.6 | 6 | 9.5 | 652.8 | 6 | 36.0 | ||||
| 4 | 40 | 110 | 312.2 | 16 | 15.3 | 1833.1 | 3 | 134.2 | ||||
| 5 | 90 | 212 | 91.1 | 16 | 3.9 | 1142.9 | 16 | 53.7 | ||||
. | . | . | Urine dGuo . | . | . | Urine inosine . | . | . | ||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Patient no. . | Dose, mg/m2 . | Dose, mg . | Amount excreted, mg . | Tmax, h . | Maximum rate, mg/h . | Amount excreted, mg . | Tmax, h . | Maximum rate, mg/h . | ||||
| 1 | 40 | 79.2 | 213.9 | 16 | 11.5 | 1151.5 | 16 | 59.8 | ||||
| 2 | 40 | 67.2 | 95.1 | 16 | 4.8 | 578.1 | 16 | 29.9 | ||||
| 3 | 40 | 64.4 | 172.6 | 6 | 9.5 | 652.8 | 6 | 36.0 | ||||
| 4 | 40 | 110 | 312.2 | 16 | 15.3 | 1833.1 | 3 | 134.2 | ||||
| 5 | 90 | 212 | 91.1 | 16 | 3.9 | 1142.9 | 16 | 53.7 | ||||