Table 4.

On target, off-tumor side effects with GPRC5D-targeting BsAb therapy

Talquetamab 400  µg/kg SC weekly (n = 30)30 Talquetamab 800  µg/kg SC biweekly (n = 44)30 Forimtamig SC (n = 57)31 
grade 1-2grade 3-4grade 1-2grade 3-4grade 1-2grade 3-4
Skin-related eventsa 67 70 82 all grade 15d 
Rash-related eventsb 47 30 16   
Nail-related eventsc 57 27 22 
Dry mouth 30 57 74e 6e 
Dysgeusia 63 NR 57 NR   
Dysphagia 37 27   
Decreased appetite 20 20   
Decreased weight 30 22   
Talquetamab 400  µg/kg SC weekly (n = 30)30 Talquetamab 800  µg/kg SC biweekly (n = 44)30 Forimtamig SC (n = 57)31 
grade 1-2grade 3-4grade 1-2grade 3-4grade 1-2grade 3-4
Skin-related eventsa 67 70 82 all grade 15d 
Rash-related eventsb 47 30 16   
Nail-related eventsc 57 27 22 
Dry mouth 30 57 74e 6e 
Dysgeusia 63 NR 57 NR   
Dysphagia 37 27   
Decreased appetite 20 20   
Decreased weight 30 22   
a

Skin-related events included asteatotic eczema, dry skin, eczema, pruritus, exfoliation, fissures, hyperpigmentation, lesions, skin toxic effects, and ulcers.

b

Rash-related events included contact dermatitis, dermatitis, erythematous rash, generalized exfoliative dermatitis, maculopapular rash, and rash.

c

Nail-related events included nail-bed disorder, discoloration, dystrophy, hypertrophy, ridging, onycholysis, and onychomadesis.

d

All skin abnormalities combined.

e

All oral toxicities combined.

NR, not reported.

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