AEs per Bearman scale
| Organ . | Grade . | |||||
|---|---|---|---|---|---|---|
| DL1: 0.4 mCi/kg (n = 4) . | DL2: 0.5 mCi/kg (n = 4) . | DL3: 0.6 mCi/kg (n = 12) . | ||||
| 1 . | 2 . | 1 . | 2 . | 1 . | 2 . | |
| Bladder | 0 | 0 | 0 | 0 | 0 | 1 |
| Cardiac | 0 | 0 | 0 | 0 | 0 | 0 |
| Central nervous system | 0 | 0 | 0 | 0 | 0 | 0 |
| GI | 0 | 2 | 2 | 0 | 5 | 0 |
| Hepatic | 1 | 0 | 0 | 0 | 0 | 0 |
| Pulmonary | 0 | 0 | 1 | 0 | 1 | 0 |
| Renal | 0 | 0 | 0 | 0 | 2 | 0 |
| Mucositis | 0 | 3 | 0 | 4 | 2 | 7 |
| Organ . | Grade . | |||||
|---|---|---|---|---|---|---|
| DL1: 0.4 mCi/kg (n = 4) . | DL2: 0.5 mCi/kg (n = 4) . | DL3: 0.6 mCi/kg (n = 12) . | ||||
| 1 . | 2 . | 1 . | 2 . | 1 . | 2 . | |
| Bladder | 0 | 0 | 0 | 0 | 0 | 1 |
| Cardiac | 0 | 0 | 0 | 0 | 0 | 0 |
| Central nervous system | 0 | 0 | 0 | 0 | 0 | 0 |
| GI | 0 | 2 | 2 | 0 | 5 | 0 |
| Hepatic | 1 | 0 | 0 | 0 | 0 | 0 |
| Pulmonary | 0 | 0 | 1 | 0 | 1 | 0 |
| Renal | 0 | 0 | 0 | 0 | 2 | 0 |
| Mucositis | 0 | 3 | 0 | 4 | 2 | 7 |
DL, dose level; GI, gastrointestinal.