IC50 of BBM and PA4 on NCI-60 panel of human tumor cell lines
| Cell line . | Panel name . | IC50 (μM) . | |
|---|---|---|---|
| BBM . | PA4 . | ||
| RPMI-8226 | Leukemia | 7.835 | 0.9439 |
| K-562 | Leukemia | 5.112 | 0.768 |
| MOLT-4 | Leukemia | 10.69 | 1.134 |
| HL-60(TB) | Leukemia | 5.976 | 0.9964 |
| CCRF-CEM | Leukemia | 11.36 | 1.007 |
| SR | Leukemia | 5.137 | 0.5188 |
| A549/ATCC | Non–small cell lung | 18.71 | 2.777 |
| NCI-H460 | Non–small cell lung | 20.53 | 1.806 |
| EKVX | Non–small cell lung | 6.376 | 1.427 |
| NCI-H522 | Non–small cell lung | 21.28 | 2.111 |
| HOP-62 | Non–small cell lung | 23.82 | 4.233 |
| NCI-H322M | Non–small cell lung | 19.96 | 3.144 |
| HOP-92 | Non–small cell lung | 12.71 | 2.792 |
| NCI-H23 | Non–small cell lung | 14.9 | 1.779 |
| NCI-H226 | Non–small cell lung | 34.55 | 3.662 |
| SW-620 | Colon | 12.41 | 1.163 |
| HT29 | Colon | 6.564 | 1.035 |
| KM12 | Colon | 17.3 | 2.158 |
| HCT-116 | Colon | 10.15 | 1.679 |
| HCT-15 | Colon | 11.04 | 1.402 |
| COLO 205 | Colon | 15.95 | 1.27 |
| HCC-2998 | Colon | 5.606 | 1.114 |
| SF-268 | CNS | 13.82 | 1.986 |
| U251 | CNS | 10.66 | 1.125 |
| SF-295 | CNS | 13.32 | 1.918 |
| SNB-19 | CNS | 16.21 | 1.866 |
| SNB-75 | CNS | 17.59 | 1.398 |
| SF-539 | CNS | 5.252 | 1.098 |
| MALME-3M | Melanoma | 9.824 | 1.423 |
| SK-MEL-2 | Melanoma | 16.01 | 1.038 |
| LOX IMVI | Melanoma | 23.04 | 1.76 |
| SK-MEL-28 | Melanoma | 15.39 | 2.467 |
| SK-MEL-5 | Melanoma | 9.896 | 1.306 |
| M14 | Melanoma | 13.06 | 1.88 |
| MDA-MB-435 | Melanoma | 13.46 | 1.819 |
| UACC-257 | Melanoma | 6.497 | 1.17 |
| UACC-62 | Melanoma | 19.23 | 1.941 |
| NCI/ADR-RES | Ovarian | 24.81 | 3.248 |
| OVCAR-3 | Ovarian | 12.26 | 2.293 |
| SK-OV-3 | Ovarian | 13.42 | 1.455 |
| IGR-OV1 | Ovarian | 29.59 | 3.384 |
| OVCAR-4 | Ovarian | 15.11 | 2.058 |
| OVCAR-5 | Ovarian | 9.876 | 1.411 |
| OVCAR-8 | Ovarian | 14.61 | 1.974 |
| ACHN | Renal | 20.78 | 2.318 |
| UO-31 | Renal | 9.613 | 1.081 |
| 786-0 | Renal | 8.476 | 1.242 |
| SN12C | Renal | 41.8 | 5.512 |
| CAKI-1 | Renal | 14.23 | 1.765 |
| TK-10 | Renal | 35.75 | 2.311 |
| RXF 393 | Renal | 16.9 | 1.916 |
| A498 | Renal | 6.971 | 1.602 |
| PC-3 | Prostate | 7.938 | 1.98 |
| DU-145 | Prostate | 27.71 | 2.732 |
| MCF7 | Breast | 9.927 | 1.784 |
| HS 578T | Breast | 12.4 | 1.339 |
| MDA-MB-468 | Breast | 10.4 | 1.528 |
| MDA-MB-231/ATCC | Breast | 14.16 | 1.265 |
| BT-549 | Breast | 8.641 | 1.208 |
| T-47D | Breast | 15.72 | 1.801 |
| FG | Pancreatic | 32.59 | 2.176 |
| BxPC3 | Pancreatic | 31.94 | 1.887 |
| Su8686 | Pancreatic | NA | 1.263 |
| Miapaca2 | Pancreatic | 20.72 | 1.122 |
| Panc1 | Pancreatic | 24.78 | 2.866 |
| CaPan2 | Pancreatic | 59.1 | 4.782 |
| Rael | Lymphoma | 5.874 | 0.6174 |
| H9 | Lymphoma | 4.668 | 0.8066 |
| Namalwa | Lymphoma | 20.71 | 2.313 |
| JB6 | Lymphoma | 2.119 | 0.7317 |
| DHL6 | Lymphoma | 15.88 | 1.018 |
| Mutu | Lymphoma | 4.636 | 0.3899 |
| Cell line . | Panel name . | IC50 (μM) . | |
|---|---|---|---|
| BBM . | PA4 . | ||
| RPMI-8226 | Leukemia | 7.835 | 0.9439 |
| K-562 | Leukemia | 5.112 | 0.768 |
| MOLT-4 | Leukemia | 10.69 | 1.134 |
| HL-60(TB) | Leukemia | 5.976 | 0.9964 |
| CCRF-CEM | Leukemia | 11.36 | 1.007 |
| SR | Leukemia | 5.137 | 0.5188 |
| A549/ATCC | Non–small cell lung | 18.71 | 2.777 |
| NCI-H460 | Non–small cell lung | 20.53 | 1.806 |
| EKVX | Non–small cell lung | 6.376 | 1.427 |
| NCI-H522 | Non–small cell lung | 21.28 | 2.111 |
| HOP-62 | Non–small cell lung | 23.82 | 4.233 |
| NCI-H322M | Non–small cell lung | 19.96 | 3.144 |
| HOP-92 | Non–small cell lung | 12.71 | 2.792 |
| NCI-H23 | Non–small cell lung | 14.9 | 1.779 |
| NCI-H226 | Non–small cell lung | 34.55 | 3.662 |
| SW-620 | Colon | 12.41 | 1.163 |
| HT29 | Colon | 6.564 | 1.035 |
| KM12 | Colon | 17.3 | 2.158 |
| HCT-116 | Colon | 10.15 | 1.679 |
| HCT-15 | Colon | 11.04 | 1.402 |
| COLO 205 | Colon | 15.95 | 1.27 |
| HCC-2998 | Colon | 5.606 | 1.114 |
| SF-268 | CNS | 13.82 | 1.986 |
| U251 | CNS | 10.66 | 1.125 |
| SF-295 | CNS | 13.32 | 1.918 |
| SNB-19 | CNS | 16.21 | 1.866 |
| SNB-75 | CNS | 17.59 | 1.398 |
| SF-539 | CNS | 5.252 | 1.098 |
| MALME-3M | Melanoma | 9.824 | 1.423 |
| SK-MEL-2 | Melanoma | 16.01 | 1.038 |
| LOX IMVI | Melanoma | 23.04 | 1.76 |
| SK-MEL-28 | Melanoma | 15.39 | 2.467 |
| SK-MEL-5 | Melanoma | 9.896 | 1.306 |
| M14 | Melanoma | 13.06 | 1.88 |
| MDA-MB-435 | Melanoma | 13.46 | 1.819 |
| UACC-257 | Melanoma | 6.497 | 1.17 |
| UACC-62 | Melanoma | 19.23 | 1.941 |
| NCI/ADR-RES | Ovarian | 24.81 | 3.248 |
| OVCAR-3 | Ovarian | 12.26 | 2.293 |
| SK-OV-3 | Ovarian | 13.42 | 1.455 |
| IGR-OV1 | Ovarian | 29.59 | 3.384 |
| OVCAR-4 | Ovarian | 15.11 | 2.058 |
| OVCAR-5 | Ovarian | 9.876 | 1.411 |
| OVCAR-8 | Ovarian | 14.61 | 1.974 |
| ACHN | Renal | 20.78 | 2.318 |
| UO-31 | Renal | 9.613 | 1.081 |
| 786-0 | Renal | 8.476 | 1.242 |
| SN12C | Renal | 41.8 | 5.512 |
| CAKI-1 | Renal | 14.23 | 1.765 |
| TK-10 | Renal | 35.75 | 2.311 |
| RXF 393 | Renal | 16.9 | 1.916 |
| A498 | Renal | 6.971 | 1.602 |
| PC-3 | Prostate | 7.938 | 1.98 |
| DU-145 | Prostate | 27.71 | 2.732 |
| MCF7 | Breast | 9.927 | 1.784 |
| HS 578T | Breast | 12.4 | 1.339 |
| MDA-MB-468 | Breast | 10.4 | 1.528 |
| MDA-MB-231/ATCC | Breast | 14.16 | 1.265 |
| BT-549 | Breast | 8.641 | 1.208 |
| T-47D | Breast | 15.72 | 1.801 |
| FG | Pancreatic | 32.59 | 2.176 |
| BxPC3 | Pancreatic | 31.94 | 1.887 |
| Su8686 | Pancreatic | NA | 1.263 |
| Miapaca2 | Pancreatic | 20.72 | 1.122 |
| Panc1 | Pancreatic | 24.78 | 2.866 |
| CaPan2 | Pancreatic | 59.1 | 4.782 |
| Rael | Lymphoma | 5.874 | 0.6174 |
| H9 | Lymphoma | 4.668 | 0.8066 |
| Namalwa | Lymphoma | 20.71 | 2.313 |
| JB6 | Lymphoma | 2.119 | 0.7317 |
| DHL6 | Lymphoma | 15.88 | 1.018 |
| Mutu | Lymphoma | 4.636 | 0.3899 |
CNS, central nervous system.