All-causality AEs occurring in >10% of all treated patients (N = 51)
AE . | Grade 1 . | Grade 2 . | Grade 3 . | Grade 4 . | ||||
---|---|---|---|---|---|---|---|---|
n . | % . | n . | % . | n . | % . | n . | % . | |
Diarrhea | 17 | 33 | 11 | 22 | 4 | 8 | 0 | 0 |
Nausea | 20 | 39 | 7 | 14 | 0 | 0 | 0 | 0 |
Fatigue | 4 | 8 | 9 | 18 | 0 | 0 | 0 | 0 |
Insomnia | 11 | 22 | 2 | 4 | 0 | 0 | 0 | 0 |
Thrombocytopenia | 4 | 8 | 3 | 6 | 4 | 8 | 2 | 4 |
Headache | 9 | 18 | 3 | 6 | 0 | 0 | 0 | 0 |
Neutropenia | 1 | 2 | 2 | 4 | 2 | 4 | 7 | 14 |
Dizziness | 8 | 16 | 2 | 4 | 0 | 0 | 0 | 0 |
Peripheral edema | 8 | 16 | 1 | 2 | 0 | 0 | 0 | 0 |
Cough | 6 | 12 | 2 | 4 | 0 | 0 | 0 | 0 |
Rash | 7 | 14 | 1 | 2 | 0 | 0 | 0 | 0 |
Rash, maculopapular | 8 | 16 | 0 | 0 | 0 | 0 | 0 | 0 |
Anemia | 1 | 2 | 4 | 8 | 2 | 4 | 0 | |
Arthralgia | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
Contusion | 7 | 14 | 0 | 0 | 0 | 0 | 0 | 0 |
Decreased appetite | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
Leukocytosis | 0 | 0 | 0 | 0 | 7 | 14 | 0 | 0 |
Myalgia | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
Pneumonia | 0 | 0 | 1 | 2 | 6 | 12 | 0 | 0 |
Pyrexia | 4 | 8 | 2 | 4 | 1 | 2 | 0 | 0 |
Upper respiratory tract infection | 4 | 8 | 3 | 6 | 0 | 0 | 0 | 0 |
Vomiting | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
AST/ALT increase | 2 | 4 | 2 | 4 | 3 | 6 | 0 | 0 |
AE . | Grade 1 . | Grade 2 . | Grade 3 . | Grade 4 . | ||||
---|---|---|---|---|---|---|---|---|
n . | % . | n . | % . | n . | % . | n . | % . | |
Diarrhea | 17 | 33 | 11 | 22 | 4 | 8 | 0 | 0 |
Nausea | 20 | 39 | 7 | 14 | 0 | 0 | 0 | 0 |
Fatigue | 4 | 8 | 9 | 18 | 0 | 0 | 0 | 0 |
Insomnia | 11 | 22 | 2 | 4 | 0 | 0 | 0 | 0 |
Thrombocytopenia | 4 | 8 | 3 | 6 | 4 | 8 | 2 | 4 |
Headache | 9 | 18 | 3 | 6 | 0 | 0 | 0 | 0 |
Neutropenia | 1 | 2 | 2 | 4 | 2 | 4 | 7 | 14 |
Dizziness | 8 | 16 | 2 | 4 | 0 | 0 | 0 | 0 |
Peripheral edema | 8 | 16 | 1 | 2 | 0 | 0 | 0 | 0 |
Cough | 6 | 12 | 2 | 4 | 0 | 0 | 0 | 0 |
Rash | 7 | 14 | 1 | 2 | 0 | 0 | 0 | 0 |
Rash, maculopapular | 8 | 16 | 0 | 0 | 0 | 0 | 0 | 0 |
Anemia | 1 | 2 | 4 | 8 | 2 | 4 | 0 | |
Arthralgia | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
Contusion | 7 | 14 | 0 | 0 | 0 | 0 | 0 | 0 |
Decreased appetite | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
Leukocytosis | 0 | 0 | 0 | 0 | 7 | 14 | 0 | 0 |
Myalgia | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
Pneumonia | 0 | 0 | 1 | 2 | 6 | 12 | 0 | 0 |
Pyrexia | 4 | 8 | 2 | 4 | 1 | 2 | 0 | 0 |
Upper respiratory tract infection | 4 | 8 | 3 | 6 | 0 | 0 | 0 | 0 |
Vomiting | 5 | 10 | 2 | 4 | 0 | 0 | 0 | 0 |
AST/ALT increase | 2 | 4 | 2 | 4 | 3 | 6 | 0 | 0 |
AST, aspartate aminotransferase.